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Publications


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Kiss and Run: Promoting Effective and Targeted Cellular Uptake of a Drug Delivery Vehicle Composed of an Integrin-Targeting Diketopiperazine Peptidomimetic and a Cell-Penetrating Peptide

Lucia Feni, Sara Parente, Clémence Robert, Silvia Gazzola, Daniela Arosio, Umberto Piarulli, Ines Neundorf
Bioconjugate Chem.2019 30, 7, 2011.
DOI: 10.1021/acs.bioconjchem.9b00292
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Synthesis and Biological Evaluation of RGD-Cryptophycin Conjugates for Targeted Drug Delivery

Adina Noémi Borbély, Eduard Figueras Agustí, Ana Martins, Simone Esposito, Giulio Auciello, Edith Monteagudo, Annalise Di Marco, Vincenzo Summa, Paola Cordella, Raffaella Perego, Isabell Kemker, Marcel Frese, Paola Gallinari, Christian Steinkühler, Norbert Sewald
Pharmaceutics  2019, 11, 151.
DOI: 10.3390/pharmaceutics11040151
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Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

Adina Borbély, Eduard Figueras, Ana Martins, Lizeth Bodero, André Raposo Moreira Dias, Paula López Rivas, Arianna Pina, Daniela Arosio, Paola Gallinari, Marcel Frese, Christian Steinkühler, Cesare Gennari, Umberto Piarulli, Norbert Sewald
ChemistryOpen 2019, 8, 737.
DOI: 10.1002/open.201900110
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Octreotide Conjugates for Tumor Targeting and Imaging

Eduard Figueras , Ana Martins , Adina Borbély, Vadim Le Joncour, Paola Cordella, Raffaella Perego, Daniela Modena, Paolo Pagani, Simone Esposito, Giulio Auciello, Marcel Frese, Paola Gallinari, Pirjo Laakkonen, Christian Steinkühler, Norbert Sewald
Pharmaceutics 2019, 11, 5, 220.
DOI: 10.3390/pharmaceutics11050220
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In Vivo Antitumor Activity of a Novel Acetazolamide-Cryptophycin Conjugate for the Treatment of Renal Cell Carcinomas

Samuele Cazzamalli, Eduard Figueras, Lilla Pethő, Adina Borbély, Christian Steinkühler, Dario Neri, Norbert Sewald
ACS Omega 2018, 3, 11, 14726.
DOI: 10.1021/acsomega.8b02350
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Novel unit B cryptophycin analogues as payloads for targeted therapy

Eduard Figueras, Adina Borbély, Mohamed Ismail, Marcel Frese, Norbert Sewald
Beilstein J. Org. Chem. 2018, 14, 1281.
DOI: 10.3762/bjoc.14.109
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Synthesis and in vitro biochemical evaluation of oxime bond-linked daunorubicin-GnRH-III conjugates developed for targeted drug delivery

Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, Viktor Farkas, László Buday, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Beilstein J. Org. Chem. 2018,14, 756.
DOI: 10.3762/bjoc.14.64
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Development of novel cyclic NGR peptide-daunomycin conjugates with dual targeting property

Andrea Angelo Pierluigi Tripodi, Szilárd Tóth, Kata Nóra Enyedi, Gitta Schlosser, Gergely Szakács, Gábor Mező
Beilstein J. Org. Chem. 2018, 14, 911.
DOI: 10.3762/bjoc.14.78
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Enhanced In Vitro Antitumor Activity of GnRH-III-Daunorubicin Bioconjugates Influenced by Sequence Modification

Sabine Schuster, Beáta Biri-Kovács, Bálint Szeder, László Buday, János Gardi, Zsuzsanna Szabó, Gábor Halmos, Gábor Mező
Pharmaceutics 2018, 10, 4, 223.
DOI: 10.3390/pharmaceutics10040223
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Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αVβ3-Integrin Ligands for Tumor Targeting

Paula López Rivas, Ivan Ranđelović, André Raposo Moreira Dias, Arianna Pina, Daniela Arosio, József Tóvári, Gábor Mező, Alberto Dal Corso, Luca Pignataro, Cesare Gennari
Eur. J. Org. Chem. 2018, 2902.
DOI: 10.1002/ejoc.201800447
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Cryptophycins: cytotoxic cyclodepsipeptides with potential for tumor targeting

Christine Weiss, Eduard Figueras, Adina N. Borbely, Norbert Sewald
J. Pept. Sci. 2017,23, 514.
DOI: 10.1002/psc.3015
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Convenient Preparation of 18F-Labeled Peptide Probes for Potential Claudin-4 PET Imaging

Lucia Feni, M. Omrane, Moritz Fischer, Boris Zlatopolskiy, Bernd Neumaier, Ines Neundorf
Pharmaceuticals  2017, 10, 99.
DOI: 10.3390/ph10040099
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The Current Role of Cell-Penetrating Peptides in Cancer Therapy.

Lucia Feni, Ines Neundorf
Peptides and Peptide-based Biomaterials and their Biomedical Applications. Advances in Experimental Medicine and Biology. 2017, 1030, 279–295.
DOI: 10.1007/978-3-319-66095-0_13



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Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αVβ3

André Raposo Moreira Dias, Arianna Pina, Alberto Dal Corso, Daniela Arosio, Laura Belvisi, Luca Pignataro, Michele Caruso, Cesare Gennari
Chem. Eur. J. 2017, 23, 14410–14415.
DOI: 10.1002/chem.201703093
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Tumor Targeting with an isoDGR-Drug Conjugate

Simone Zanella, Simona Angerani, Arianna Pina, Paula López Rivas, Clelia Giannini, Silvia Panzeri, Daniela Arosio, Michele Caruso, Fabio Gasparri, Ivan Fraietta, Clara Albanese, Aurelio Marsiglio, Luca Pignataro, Laura Belvisi, Umberto Piarulli, Cesare Gennari
Chem. Eur. J. 2017, 23, 7910–7914.
DOI: 10.1002/chem.201701844
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Characterization of a Cell-Penetrating Peptide with Potential Anticancer Activity

Anja Gronewold, Mareike Horn, Ivan Ranđelović, József Tóvári, Sergio Muñoz Vázquez, Klaus Schomäcker, Ines Neundorf
ChemMedChem 2017, 12, 42–49.
DOI: 10.1002/cmdc.201600498
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